产品说明
一般描述
A potent and competitive inhibitor of protein kinase A (Ki = 1.7 nM).
A potent and competitive inhibitor of PKA (Ki = 1.7 nM).
包装
1 mg in Plastic ampoule
Yes
生化/生理作用
Product does not compete with ATP.
Primary Target
PKA
Target Ki: 1.7 nM against protein kinase A
Reversible: no
Cell permeable: no
警告
Toxicity: Standard Handling (A)
序列
H-Thr-Tyr-Ala-Asp-Phe-Ile-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-Ile-NH₂
外形
Supplied as a trifluoroacetate salt.
重悬
Following initial thaw, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
其他说明
Glass, D.B., et al. 1989. J. Biol. Chem. 264, 8802.
Kemp, B.E., et al. 1988. Methods Enzymol.159, 173.
法律信息
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
基本信息
经验(实验)分子式 | C80H130N28O24 |
分子量 | 1868.06 |
MDL编号 | MFCD00133792 |
产品性质
质量水平 | 100 |
测定 | ≥97% (HPLC) |
形式 | solid |
manufacturer/tradename | Calbiochem® |
储存条件 | OK to freeze desiccated (hygroscopic) |
溶解性 | water: 1 mg/mL |
运输 | ambient |
储存温度 | −20℃ |
安全信息
储存分类代码 | 11 - Combustible Solids |
WGK | WGK 3 |
闪点(F) | Not applicable |
闪点(C) | Not applicable |