产品说明
一般描述
Note: this peptide forms cyclic isomers.
Lysinal analog of Leupeptin (Cat. No. 108975). A more potent inhibitor of cathepsin B (IC50 = 4 nM) than of leupeptin (IC50 = 310 nM). Note: this peptide forms cyclic isomers.
A more active lysinal analog of Leupeptin (Cat. No. 108975). A more potent inhibitor of cathepsin B (IC50 = 4 nM) compared to leupeptin (IC50 = 310 nM).
包装
1 mg in Plastic ampoule
生化/生理作用
Product does not compete with ATP.
Primary Target
cathepsin B
Reversible: no
Target IC50: 4 nM against cathepsin B
Cell permeable: no
警告
Toxicity: Standard Handling (A)
序列
Ac-Leu-Val-lysinal
重悬
Following reconstitution aliquot and freeze (-70°C). Stock solutions are stable for up to 1 month at -70°C.
其他说明
McConnell, R.M., et al. 1993. J. Med. Chem. 36, 1084.
法律信息
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
基本信息
| 经验(实验)分子式 | C19H36N4O4 |
| 分子量 | 384.51 |
产品性质
| 质量水平 | 100 |
| 测定 | ≥95% (HPLC) |
| 形式 | solid |
| manufacturer/tradename | Calbiochem® |
| 储存条件 | OK to freeze |
| 颜色 | white |
| 溶解性 | water: 1 mg/mL |
| 运输 | ambient |
| 储存温度 | −70℃ |
安全信息
| 储存分类代码 | 11 - Combustible Solids |
| WGK | WGK 1 |
| 闪点(F) | Not applicable |
| 闪点(C) | Not applicable |
