产品说明
一般描述
Highly specific cell-permeable, reversible, and ATP-competitive inhibitor of protein kinase G (Ki = 234 nM). Inhibits protein kinase C (Ki = 4.0 µM) and protein kinase A (Ki >10.0 µM) at higher concentrations.
Highly specific, cell-permeable, reversible, and ATP-competitive inhibitor of protein kinase G (Ki = 234 nM).
包装
50, 100 μg in Plastic ampoule
生化/生理作用
Cell permeable: yes
Primary Target
PKG
Product competes with ATP.
Reversible: yes
Target Ki: 234 nM against protein kinase G
警告
Toxicity: Standard Handling (A)
制备说明
Further dilute with aqueous buffers just prior to use.
重悬
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
其他说明
Grider, J.R. 1993. Am. J. Physiol.264, G334.
法律信息
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
基本信息
| 经验(实验)分子式 | C29H25N3O5 |
| 分子量 | 495.53 |
| MDL编号 | MFCD09878278 |
产品性质
| 质量水平 | 100 |
| 测定 | ≥98% (HPLC) |
| 形式 | solid |
| manufacturer/tradename | Calbiochem® |
| 储存条件 | OK to freeze protect from light |
| 颜色 | white |
| 溶解性 | DMSO: 1 mg/mL DMF: soluble |
| 运输 | ambient |
| 储存温度 | −20℃ |
| InChI | 1S/C29H25N3O5/c1-28-29(36-4,27(34)35-3)13-20(37-28)31-18-11-7-5-9-15(18)22-23-17(14-30(2)26(23)33)21-16-10-6-8-12-19(16)32(28)25(21)24(22)31/h5-12,20H,13-14H2,1-4H3/t20-,28+,29+/m1/s1 |
| InChI key | QTYMDECKVKSGSM-YMUMJAELSA-N |
安全信息
| 储存分类代码 | 11 - Combustible Solids |
| WGK | WGK 3 |
| 闪点(F) | Not applicable |
| 闪点(C) | Not applicable |
