- 货号:5.31126CAS:包装:25 mg分子式:C10H8N2OS纯度规格:A cell-permeable. Reversible, selective inhibitor of the growth of malignant peripheral nerve sheath tumors (EC50 = 439 nM, 754 nM, and 1.0 μM in S462, SNF96.2, and sMPNST cells).分子量:204.25
- 货号:5.09884CAS:包装:10 mg分子式:C47H75N9O14纯度规格:A cell-permeable myristoylated hexapeptide that selectively inhibits integrin outside-in signaling without affecting inside-out signaling. Blocks the interaction of Gα3 and integrin β3 subunit.分子量:990.15
- 货号:5.32813CAS:包装:10 mg分子式:C20H18ClF6N3O2纯度规格:A cell-permeable compound that selectively downregulates the expression of p21 (~10 μM), independent of p53.expression, at either transcription or post-transcriptional level.分子量:481.82
- 货号:5.08957CAS:包装:5 mg分子式:C22H20ClN3O2纯度规格:A cell-permeable, highly potent and selective inhibitor of phosphodiesterase 5 (PDEV; IC50 = 270 pM).分子量:393.87
- 货号:5.05206CAS:包装:10 mg分子式:C15H13N3OS2纯度规格:A rhodanine-derived, reversible, photoactivated, TrpA1-selective channel activator.分子量:315.41
- 货号:5.31091CAS:1243244-14-5包装:5 mg分子式:C23H20N6O纯度规格:A cell-permeable inhibitor of Wnt secretion from L-cell Wnt1/2/3/3a/6/7a/9a transfectants (IC50 from 50 pM to 1.1 nM).分子量:396.44
- 货号:5.06074CAS:包装:10 MG分子式:C16H19N3O2 · xHCl纯度规格:分子量:285.34 (free base basis)
- 货号:5.06046CAS:包装:10 mg分子式:C17H15NO5纯度规格:A cell-permeable, selective inhibitor of protein arginine methyltransferase 1 (PRMT1; IC50 = 9.5 μM).分子量:313.30
- 货号:5.05763CAS:64924-67-0包装:10 mg分子式:C16H17BrClN3O3 · xHBr纯度规格:A cell-permeable racemic mixture of Halofuginone that inhibits of prolyl-tRNA synthetase.分子量:414.68 (free base basis)
- 货号:5.06188CAS:79559-97-0包装:10 MG分子式:C17H17Cl2N · xHCl纯度规格:分子量:306.23 (free base basis)
- 货号:5.09708CAS:127729-35-5包装:10 mg分子式:C4H12NO2P纯度规格:A highly potent agonist of GABAB receptor. Shown to be about 10-times more potent than baclofen.分子量:137.12
- 货号:5.30236CAS:包装:10 mg分子式:C26H38N2O · 2HCl纯度规格:A cell-permeable inhibitor of SKP2-dependent p27Kip1 ubiquitination. Selectively induces the accumulation SCFSKP2 substrates in multiple myeloma RPMI 8226 cells.分子量:467.51
- 货号:5.08512CAS:203460-30-4包装:10 μg分子式:C192H274N52O60S7纯度规格:A peptidyl toxin from venom of African tarantula, Hysterocrates gigas that acts as a high affinity, reversible blocker of Cav2.3 (α1E, R-type) channels (IC50 = 15-30 nM).分子量:4495.00
- 货号:5.09106CAS:包装:10 mg分子式:C18H24N2O3S纯度规格:A cell permeable, selective, sphingosine competitive inhibitor of spingosine Kinase -2 (IC50 = 4.3 μM).分子量:348.46
- 货号:5.30487CAS:827022-32-2包装:5 mg分子式:C24H29N7O2 · xHCl纯度规格:A cell-permeable, brain permeant, potent, reversible, ATP competitive inhibitor of Cdk4 and Cdk6 (IC50 = 11, 9, and 15 nM for Cdk4/D1, Cdk4/D3 and Cdk6/D2, respectively).分子量:447.53 (free base basis)
- 货号:5.31889CAS:1441190-66-4包装:500 μG分子式:纯度规格:分子量:
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